nitenpyram 🐶 Veterinary Use | Indications/Contra | FAERs-F | FAERs-M | Orange Bk | BioActivity |
| Stem definition | Drug id | CAS RN |
|---|---|---|
| 5587 | 150824-47-8 |
Description:
| Molecule | Description |
|---|---|
|
Synonyms:
|
A nitromethylene neonicotinoid insecticide
|
Drug dosage:
None
ADMET properties:
None
Approvals:
| Date | Agency | Company | Orphan |
|---|---|---|---|
| None | FDA |
FDA Adverse Event Reporting System (Female)
None
FDA Adverse Event Reporting System (Male)
None
FDA Adverse Event Reporting System (Geriatric)
None
FDA Adverse Event Reporting System (Pediatric)
None
Pharmacologic Action:
| Source | Code | Description |
|---|---|---|
| MeSH PA | D007306 | Insecticides |
| MeSH PA | D010575 | Pesticides |
Drug Use | Suggest Off label Use Form| |View source of the data|
None
🐶 Veterinary Drug Use
| Species | Use | Relation |
|---|---|---|
| Cats | Flea infestations | Indication |
| Dogs | Flea infestations | Indication |
🐶 Veterinary products
| Product | Applicant | Ingredients |
|---|---|---|
| CAPSTAR | Sergeant?s Pet Care Products LLC | 1 |
| Sentinel Flavor Tabs and Capstar Flea Management System | Intervet Inc. | 3 |
| Program Flavor Tabs and Capstar Flea Management System | Elanco US Inc. | 2 |
Acid dissociation constants calculated using MoKa v3.0.0
None
Orange Book patent data (new drug applications)
None
Orange Book exclusivity data (new drug applications)
None
Bioactivity Summary:
| Target | Class | Pharos | UniProt | Action | Type | Activity value (-log[M]) | Mechanism action | Bioact source | MoA source |
|---|---|---|---|---|---|---|---|---|---|
| Acetylcholine receptor subunit beta-like 2 | Ion channel | IC50 | 7.96 | CHEMBL |
External reference:
| ID | Source |
|---|---|
| CHEBI:39170 | CHEBI |
| CHEMBL259728 | ChEMBL_ID |
| C464843 | MESH_SUPPLEMENTAL_RECORD_UI |
| DB11438 | DRUGBANK_ID |
| C1143123 | UMLSCUI |
| C18511 | KEGG_DRUG |
| 3034287 | PUBCHEM_CID |
| 341379 | RXNORM |
| 3A837VZ81Y | UNII |
Pharmaceutical products:
None